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Target
Dual specificity protein phosphatase 26
Ligand
BDBM50087879
Substrate
n/a
Meas. Tech.
ChEMBL_929798 (CHEMBL3068773)
IC50
16700±n/a nM
Citation
  TBA Med Chem Res 22:3905-3910 (2013)    Article 
Target
Name:
Dual specificity protein phosphatase 26
Synonyms:
3.1.3.16 | 3.1.3.48 | DSP-4 | DUS26_HUMAN | DUSP24 | DUSP26 | Dual specificity phosphatase SKRP3 | Dual specificity protein phosphatase 26 | LDP-4 | LDP4 | Low-molecular-mass dual-specificity phosphatase 4 | MAP kinase phosphatase 8 | MKP-8 | MKP8 | Mitogen-activated protein kinase phosphatase 8 | NATA1 | Novel amplified gene in thyroid anaplastic cancer | SKRP3
Type:
PROTEIN
Mol. Mass.:
23957.92
Organism:
Homo sapiens
Description:
ChEMBL_105561
Residue:
211
Sequence:
MCPGNWLWASMTFMARFSRSSSRSPVRTRGTLEEMPTVQHPFLNVFELERLLYTGKTACNHADEVWPGLYLGDQDMANNRRELRRLGITHVLNASHSRWRGTPEAYEGLGIRYLGVEAHDSPAFDMSIHFQTAADFIHRALSQPGGKILVHCAVGVSRSATLVLAYLMLYHHLTLVEAIKKVKDHRGIIPNRGFLRQLLALDRRLRQGLEA
  
Inhibitor
Name:
BDBM50087879
Synonyms:
CHEMBL472004 | NSC-87877
Type:
Small organic molecule
Emp. Form.:
C19H13N3O7S2
Mol. Mass.:
459.452
SMILES:
Oc1c(cc(c2cccnc12)S(O)(=O)=O)\N=N\c1ccc2cc(ccc2c1)S(O)(=O)=O
Structure:
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