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Target
Mu-type opioid receptor
Ligand
BDBM50453515
Substrate
n/a
Meas. Tech.
ChEMBL_138745 (CHEMBL747918)
Ki
310±n/a nM
Citation
 Mosberg, HI; Lomize, AL; Wang, C; Kroona, H; Heyl, DL; Sobczyk-Kojiro, K; Ma, W; Mousigian, C; Porreca, F Development of a model for the delta opioid receptor pharmacophore. 1. Conformationally restricted Tyr1 replacements in the cyclic delta receptor selective tetrapeptide Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13). J Med Chem 37:4371-83 (1995) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50453515
Synonyms:
CHEMBL2111933
Type:
Small organic molecule
Emp. Form.:
C28H34N4O6S2
Mol. Mass.:
586.723
SMILES:
CC1(C)SSC[C@H](NC(=O)[C@@]2(N)CCc3cc(O)ccc3C2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H]1C(O)=O
Structure:
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