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Target
D(3) dopamine receptor
Ligand
BDBM50054337
Substrate
n/a
Meas. Tech.
ChEMBL_62275 (CHEMBL674410)
Ki
23.8±n/a nM
Citation
 Malmberg, A; Höök, BB; Johansson, AM; Hacksell, U Novel (R)-2-amino-5-fluorotetralins: dopaminergic antagonists and inverse agonists. J Med Chem 39:4421-9 (1996) [PubMed]  Article 
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3
Type:
n/a
Mol. Mass.:
44243.43
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
400
Sequence:
MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTVCSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQQTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRKLSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHVSPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
  
Inhibitor
Name:
BDBM50054337
Synonyms:
Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine | CHEMBL65847
Type:
Small organic molecule
Emp. Form.:
C20H24FN
Mol. Mass.:
297.4097
SMILES:
CCCN(Cc1ccccc1)[C@@H]1CCc2c(F)cccc2C1
Structure:
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