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Target
Potassium channel subfamily K member 17
Ligand
BDBM50123519
Substrate
n/a
Meas. Tech.
ChEMBL_1822388 (CHEMBL4322152)
IC50
8100±n/a nM
Citation
Bedoya, M; Rinné, S; Kiper, AK; Decher, N; González, W; Ramírez, D TASK Channels Pharmacology: New Challenges in Drug Design. J Med Chem 62:10044-10058 (2019) [PubMed] Article
More Info.:
Target
Name:
Potassium channel subfamily K member 17
Synonyms:
2P domain potassium channel Talk-2 | Acid-sensitive potassium channel protein TASK-4 | KCNK17 | KCNKH_HUMAN | Potassium channel subfamily K member 17 | TALK-2 | TALK2 | TASK4 | TASK4 | TWIK-related acid-sensitive K(+) channel 4 | TWIK-related alkaline pH-activated K(+) channel 2
Type:
PROTEIN
Mol. Mass.:
36902.23
Organism:
Homo sapiens
Description:
ChEMBL_119183
Residue:
332
Sequence:
MYRPRARAAPEGRVRGCAVPSTVLLLLAYLAYLALGTGVFWTLEGRAAQDSSRSFQRDKWELLQNFTCLDRPALDSLIRDVVQAYKNGASLLSNTTSMGRWELVGSFFFSVSTITTIGYGNLSPNTMAARLFCIFFALVGIPLNLVVLNRLGHLMQQGVNHWASRLGGTWQDPDKARWLAGSGALLSGLLLFLLLPPLLFSHMEGWSYTEGFYFAFITLSTVGFGDYVIGMNPSQRYPLWYKNMVSLWILFGMAWLALIIKLILSQLETPGRVCSCCHHSSKEDFKSQSWRQGPDREPESHSPQQGCYPEGPMGIIQHLEPSAHAAGCGKDS