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Target
Cannabinoid receptor 2
Ligand
BDBM50511104
Substrate
n/a
Meas. Tech.
ChEMBL_1843636 (CHEMBL4344063)
Ki
51±n/a nM
Citation
 Linciano, P; Citti, C; Luongo, L; Belardo, C; Maione, S; Vandelli, MA; Forni, F; Gigli, G; Laganą, A; Montone, CM; Cannazza, G Isolation of a High-Affinity Cannabinoid for the Human CB1 Receptor from a Medicinal  J Nat Prod 83:88-98 (2020) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM50511104
Synonyms:
CHEMBL4437290
Type:
Small organic molecule
Emp. Form.:
C20H28O2
Mol. Mass.:
300.4351
SMILES:
[H][C@@]12C=C(C)CC[C@@]1([H])C(C)(C)Oc1cc(CCCC)cc(O)c21 |r,t:2|
Structure:
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