Reaction Details Report a problem with these data
Target
Cyclin-dependent kinase 3
Ligand
BDBM50511931
Substrate
n/a
Meas. Tech.
ChEMBL_1846252 (CHEMBL4346793)
IC50
29±n/a nM
Citation
Tadesse, S; Caldon, EC; Tilley, W; Wang, S Cyclin-Dependent Kinase 2 Inhibitors in Cancer Therapy: An Update. J Med Chem 62:4233-4251 (2019) [PubMed] Article
More Info.:
Target
Name:
Cyclin-dependent kinase 3
Synonyms:
CDK3 | CDK3/Cyclin E | CDK3_HUMAN | CDKN3 | Cyclin-dependent kinase 3 | Cyclin-dependent kinase 3 (CDK3)
Type:
Enzyme
Mol. Mass.:
35053.88
Organism:
Homo sapiens (Human)
Description:
Q00526
Residue:
305
Sequence:
MDMFQKVEKIGEGTYGVVYKAKNRETGQLVALKKIRLDLEMEGVPSTAIREISLLKELKHPNIVRLLDVVHNERKLYLVFEFLSQDLKKYMDSTPGSELPLHLIKSYLFQLLQGVSFCHSHRVIHRDLKPQNLLINELGAIKLADFGLARAFGVPLRTYTHEVVTLWYRAPEILLGSKFYTTAVDIWSIGCIFAEMVTRKALFPGDSEIDQLFRIFRMLGTPSEDTWPGVTQLPDYKGSFPKWTRKGLEEIVPNLEPEGRDLLMQLLQYDPSQRITAKTALAHPYFSSPEPSPAARQYVLQRFRH