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Target
Chromodomain Y-like protein 2
Ligand
BDBM50515913
Substrate
n/a
Meas. Tech.
ChEMBL_1862778 (CHEMBL4363634)
Kd
14100±n/a nM
Citation
 Yang, L; Liu, Y; Fan, M; Zhu, G; Jin, H; Liang, J; Liu, Z; Huang, Z; Zhang, L Identification and characterization of benzo[d]oxazol-2(3H)-one derivatives as the first potent and selective small-molecule inhibitors of chromodomain protein CDYL. Eur J Med Chem 182:0 (2019) [PubMed]  Article 
Target
Name:
Chromodomain Y-like protein 2
Synonyms:
CDY-like 2 | CDYL2 | CDYL2_HUMAN | Chromodomain Y-like protein 2
Type:
PROTEIN
Mol. Mass.:
56517.92
Organism:
Homo sapiens (Human)
Description:
ChEMBL_116982
Residue:
506
Sequence:
MASGDLYEVERIVDKRKNKKGKWEYLIRWKGYGSTEDTWEPEHHLLHCEEFIDEFNGLHMSKDKRIKSGKQSSTSKLLRDSRGPSVEKLSHRPSDPGKSKGTSHKRKRINPPLAKPKKGYSGKPSSGGDRATKTVSYRTTPSGLQIMPLKKSQNGMENGDAGSEKDERHFGNGSHQPGLDLNDHVGEQDMGECDVNHATLAENGLGSALTNGGLNLHSPVKRKLEAEKDYVFDKRLRYSVRQNESNCRFRDIVVRKEEGFTHILLSSQTSDNNALTPEIMKEVRRALCNAATDDSKLLLLSAVGSVFCSGLDYSYLIGRLSSDRRKESTRIAEAIRDFVKAFIQFKKPIVVAINGPALGLGASILPLCDIVWASEKAWFQTPYATIRLTPAGCSSYTFPQILGVALANEMLFCGRKLTAQEACSRGLVSQVFWPTTFSQEVMLRVKEMASCSAVVLEESKCLVRSFLKSVLEDVNEKECLMLKQLWSSSKGLDSLFSYLQDKIYEV
  
Inhibitor
Name:
BDBM50515913
Synonyms:
CHEMBL4448020
Type:
Small organic molecule
Emp. Form.:
C17H11FN2O3
Mol. Mass.:
310.2792
SMILES:
Fc1ccc2oc(=O)n(CC(=O)c3c[nH]c4ccccc34)c2c1
Structure:
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