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Target
Chromodomain Y-like protein 2
Ligand
BDBM50515915
Substrate
n/a
Meas. Tech.
ChEMBL_1862778 (CHEMBL4363634)
Kd
57800±n/a nM
Citation
 Yang, L; Liu, Y; Fan, M; Zhu, G; Jin, H; Liang, J; Liu, Z; Huang, Z; Zhang, L Identification and characterization of benzo[d]oxazol-2(3H)-one derivatives as the first potent and selective small-molecule inhibitors of chromodomain protein CDYL. Eur J Med Chem 182:0 (2019) [PubMed]  Article 
Target
Name:
Chromodomain Y-like protein 2
Synonyms:
CDY-like 2 | CDYL2 | CDYL2_HUMAN | Chromodomain Y-like protein 2
Type:
PROTEIN
Mol. Mass.:
56517.92
Organism:
Homo sapiens (Human)
Description:
ChEMBL_116982
Residue:
506
Sequence:
MASGDLYEVERIVDKRKNKKGKWEYLIRWKGYGSTEDTWEPEHHLLHCEEFIDEFNGLHMSKDKRIKSGKQSSTSKLLRDSRGPSVEKLSHRPSDPGKSKGTSHKRKRINPPLAKPKKGYSGKPSSGGDRATKTVSYRTTPSGLQIMPLKKSQNGMENGDAGSEKDERHFGNGSHQPGLDLNDHVGEQDMGECDVNHATLAENGLGSALTNGGLNLHSPVKRKLEAEKDYVFDKRLRYSVRQNESNCRFRDIVVRKEEGFTHILLSSQTSDNNALTPEIMKEVRRALCNAATDDSKLLLLSAVGSVFCSGLDYSYLIGRLSSDRRKESTRIAEAIRDFVKAFIQFKKPIVVAINGPALGLGASILPLCDIVWASEKAWFQTPYATIRLTPAGCSSYTFPQILGVALANEMLFCGRKLTAQEACSRGLVSQVFWPTTFSQEVMLRVKEMASCSAVVLEESKCLVRSFLKSVLEDVNEKECLMLKQLWSSSKGLDSLFSYLQDKIYEV
  
Inhibitor
Name:
BDBM50515915
Synonyms:
CHEMBL4434825
Type:
Small organic molecule
Emp. Form.:
C19H12N2O4S
Mol. Mass.:
364.375
SMILES:
[O-][N+](=O)c1ccc2n(CC(=O)c3ccc4ccccc4c3)c(=O)sc2c1
Structure:
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