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Target
Cholecystokinin receptor type A
Ligand
BDBM50073050
Substrate
n/a
Meas. Tech.
ChEMBL_50033 (CHEMBL666753)
Ki
7±n/a nM
Citation
 Kordik, CP; Reitz, AB Pharmacological treatment of obesity: therapeutic strategies. J Med Chem 42:181-201 (1999) [PubMed]  Article 
Target
Name:
Cholecystokinin receptor type A
Synonyms:
CCK-A receptor | CCK-AR | CCK1-R | CCKAR_MOUSE | Cckar | Cholecystokinin A receptor | Cholecystokinin receptor | Cholecystokinin receptor type A | Cholecystokinin-1 receptor
Type:
PROTEIN
Mol. Mass.:
48454.29
Organism:
Mus musculus
Description:
ChEMBL_40042
Residue:
436
Sequence:
MDVVDSLLMNGSNITPPCELGLENETLFCLDQPQPSKEWQSAVQILLYSFIFLLSVLGNTLVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPNLLKDFIFGSAVCKTTTYFMGTSVSVSTFNLVAISLERYGAICRPLQSRVWQTKSHALKVIAATWCLSFTIMTPYPIYSNLVPFTKNNNQTANMCRFLLPSDAMQQSWQTFLLLILFLIPGVVMVVAYGLISLELYQGIKFDASQKKSAKEKRLSSGGGGGGGSSSSRYEDSDGCYLQKSRPPRKLELQQLSTSSSGGRINRIRSSGSAANLIAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAEKHLSGTPISFILLLSYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGPTGVRGEVGEEEDGRTIRASLSRYSYSHMSTSAPPH
  
Inhibitor
Name:
BDBM50073050
Synonyms:
(S)-1-(3-Amino-pentanoyl)-2,3-dihydro-1H-indole-2-carboxylic acid butylamide | CHEMBL61498
Type:
Small organic molecule
Emp. Form.:
C18H27N3O2
Mol. Mass.:
317.4259
SMILES:
CCCCNC(=O)[C@@H]1Cc2ccccc2N1C(=O)CC(N)CC
Structure:
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