Reaction Details Report a problem with these data
Target
Spindlin-3
Ligand
BDBM50519514
Substrate
n/a
Meas. Tech.
ChEMBL_1875899 (CHEMBL4377293)
Kd
170±n/a nM
Citation
Xiong, Y; Greschik, H; Johansson, C; Seifert, L; Bacher, J; Park, KS; Babault, N; Martini, M; Fagan, V; Li, F; Chau, I; Christott, T; Dilworth, D; Barsyte-Lovejoy, D; Vedadi, M; Arrowsmith, CH; Brennan, P; Fedorov, O; Jung, M; Farnie, G; Liu, J; Oppermann, U; Schüle, R; Jin, J Discovery of a Potent and Selective Fragment-like Inhibitor of Methyllysine Reader Protein Spindlin 1 (SPIN1). J Med Chem 62:8996-9007 (2019) [PubMed] Article
More Info.:
Target
Name:
Spindlin-3
Synonyms:
SPIN-3 | SPIN3 | SPIN3_HUMAN | Spindlin-3 | Spindlin-like protein 3
Type:
PROTEIN
Mol. Mass.:
29208.24
Organism:
Homo sapiens
Description:
ChEMBL_119075
Residue:
258
Sequence:
MKTPFGKAAAGQRSRTGAGHGSVSVTMIKRKAAHKKHRSRPTSQPRGNIVGCRIQHGWKDGDEPLTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELHRDERVSSLEVLPNRVASSRISDTHLAEIMVGKAVEHIFETEEGSKNEWRGMVLAQAPVMNTWFYITYEKDPVLYMYQLLDDYKDGDLRILQDSNDSPLAEREPGEVIDSLVGKQVEYAKDDGSKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLVKTS