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Target
Target of rapamycin complex subunit LST8
Ligand
BDBM50529396
Substrate
n/a
Meas. Tech.
ChEMBL_1908592 (CHEMBL4410950)
IC50
30±n/a nM
Citation
Ouvry, G; Clary, L; Tomas, L; Aurelly, M; Bonnary, L; Borde, E; Bouix-Peter, C; Chantalat, L; Defoin-Platel, C; Deret, S; Forissier, M; Harris, CS; Isabet, T; Lamy, L; Luzy, AP; Pascau, J; Soulet, C; Taddei, A; Taquet, N; Thoreau, E; Varvier, E; Vial, E; Hennequin, LF Impact of Minor Structural Modifications on Properties of a Series of mTOR Inhibitors. ACS Med Chem Lett 10:1561-1567 (2019) [PubMed] Article
More Info.:
Target
Name:
Target of rapamycin complex subunit LST8
Synonyms:
G protein beta subunit-like | GBL | Gable | LST8 | LST8_HUMAN | MLST8 | Mammalian lethal with SEC13 protein 8 | Protein GbetaL | TORC subunit LST8 | Target of rapamycin complex subunit LST8
Type:
PROTEIN
Mol. Mass.:
35871.25
Organism:
Homo sapiens
Description:
ChEMBL_118692
Residue:
326
Sequence:
MNTSPGTVGSDPVILATAGYDHTVRFWQAHSGICTRTVQHQDSQVNALEVTPDRSMIAAAGYQHIRMYDLNSNNPNPIISYDGVNKNIASVGFHEDGRWMYTGGEDCTARIWDLRSRNLQCQRIFQVNAPINCVCLHPNQAELIVGDQSGAIHIWDLKTDHNEQLIPEPEVSITSAHIDPDASYMAAVNSTGNCYVWNLTGGIGDEVTQLIPKTKIPAHTRYALQCRFSPDSTLLATCSADQTCKIWRTSNFSLMTELSIKSGNPGESSRGWMWGCAFSGDSQYIVTASSDNLARLWCVETGEIKREYGGHQKAVVCLAFNDSVLG