Reaction Details Report a problem with these data
Target
2',5'-phosphodiesterase 12
Ligand
BDBM50532283
Substrate
n/a
Meas. Tech.
ChEMBL_1922385 (CHEMBL4425341)
IC50
0.800000±n/a nM
Citation
Franzini, RM; Randolph, C Chemical Space of DNA-Encoded Libraries. J Med Chem 59:6629-44 (2016) [PubMed] Article
More Info.:
Target
Name:
2',5'-phosphodiesterase 12
Synonyms:
2-PDE | 3.1.13.4 | 3.1.4.- | Mitochondrial deadenylase | PDE12 | PDE12_HUMAN
Type:
PROTEIN
Mol. Mass.:
67351.24
Organism:
Homo sapiens
Description:
ChEMBL_119092
Residue:
609
Sequence:
MWRLPGARAALRVIRTAVEKLSRAEAGSQTAAGAMERAVVRCVPSEPKLSLSFALADGSHKNMQRDQSEPLGRVLSRIATNALKGHAKAAAAKKSRKSRPNASGGAACSGPGPEPAVFCEPVVKLYYREEAVAEDVLNVDAWQDGAVLQIGDVKYKVERNPPAFTELQLPRYIMAGFPVCPKLSLEFGDPASSLFRWYKEAKPGAAEPEVGVPSSLSPSSPSSSWTETDVEERVYTPSNADIGLRLKLHCTPGDGQRFGHSRELESVCVVEAGPGTCTFDHRHLYTKKVTEDALIRTVSYNILADTYAQTEFSRTVLYPYCAPYALELDYRQNLIQKELTGYNADVICLQEVDRAVFSDSLVPALEAFGLEGVFRIKQHEGLATFYRKSKFSLLSQHDISFYEALESDPLHKELLEKLVLYPSAQEKVLQRSSVLQVSVLQSTKDSSKRICVANTHLYWHPKGGYIRLIQMAVALAHIRHVSCDLYPGIPVIFCGDFNSTPSTGMYHFVINGSIPEDHEDWASNGEEERCNMSLTHFFKLKSACGEPAYTNYVGGFHGCLDYIFIDLNALEVEQVIPLPSHEEVTTHQALPSVSHPSDHIALVCDLKWK