Reaction Details Report a problem with these data
Target
Chromobox protein homolog 6
Ligand
BDBM50157430
Substrate
n/a
Meas. Tech.
ChEMBL_1977191 (CHEMBL4610326)
IC50
16000±n/a nM
Citation
Milosevich, N; McFarlane, J; Gignac, MC; Li, J; Brown, TM; Wilson, CR; Devorkin, L; Croft, CS; Hof, R; Paci, I; Lum, JJ; Hof, F Pan-specific and partially selective dye-labeled peptidic inhibitors of the polycomb paralog proteins. Bioorg Med Chem 28:0 (2020) [PubMed] Article
More Info.:
Target
Name:
Chromobox protein homolog 6
Synonyms:
CBX6 | CBX6_HUMAN | Chromobox protein homolog 6
Type:
PROTEIN
Mol. Mass.:
43924.51
Organism:
Homo sapiens (Human)
Description:
ChEMBL_116765
Residue:
412
Sequence:
MELSAVGERVFAAESIIKRRIRKGRIEYLVKWKGWAIKYSTWEPEENILDSRLIAAFEQKERERELYGPKKRGPKPKTFLLKARAQAEALRISDVHFSVKPSASASSPKLHSSAAVHRLKKDIRRCHRMSRRPLPRPDPQGGSPGLRPPISPFSETVRIINRKVKPREPKRNRIILNLKVIDKGAGGGGAGQGAGALARPKVPSRNRVIGKSKKFSESVLRTQIRHMKFGAFALYKPPPAPLVAPSPGKAEASAPGPGLLLAAPAAPYDARSSGSSGCPSPTPQSSDPDDTPPKLLPETVSPSAPSWREPEVLDLSLPPESAATSKRAPPEVTAAAGPAPPTAPEPAGASSEPEAGDWRPEMSPCSNVVVTDVTSNLLTVTIKEFCNPEDFEKVAAGVAGAAGGGGSIGASK