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Target
G-protein coupled receptor 84
Ligand
BDBM50556779
Substrate
n/a
Meas. Tech.
ChEMBL_2057184 (CHEMBL4712185)
IC50
68±n/a nM
Citation
 Chen, LH; Zhang, Q; Xie, X; Nan, FJ Modulation of the G-Protein-Coupled Receptor 84 (GPR84) by Agonists and Antagonists. J Med Chem 63:15399-15409 (2020) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 84
Synonyms:
G-protein coupled receptor 84 | GPR84_MOUSE | Gpr84
Type:
PROTEIN
Mol. Mass.:
43740.69
Organism:
Mus musculus
Description:
ChEMBL_119136
Residue:
396
Sequence:
MWNSSDANFSCYHESVLGYRYFAVIWGVAVAVTGTVGNVLTLLALAIRPKLRTRFNLLIANLTLADLLYCTLLQPFSVDTYLHLHWRTGAVFCRIFGLLLFTSNSVSILTLCLIALGRYLLIAHPKLFPQVFSAKGIVLALVGSWVVGVTSFAPLWNVFVLVPVVCTCSFDRMRGRPYTTILMGIYFVLGLSSVGVFYCLIHRQVKRAARALDQYGLHQASIRSHQVAGTQEAMPGHFQELDSGVASRGPSEGISSEPVSAATTQTLEGDSSEAGGQGIRKAAQQIAERSLPEVHRKPRETAGARRATDAPSEFGKVTRMCFAVFLCFALSYIPFLLLNILDARGRAPRVVHMVAANLTWLNSCINPVLYAAMNRQFRHAYGSILKRGPQSFRRFH
  
Inhibitor
Name:
BDBM50556779
Synonyms:
CHEMBL3715656
Type:
Small organic molecule
Emp. Form.:
C26H25N3O4
Mol. Mass.:
443.4944
SMILES:
O=c1nc(OCC2COCCO2)cc2-c3ccc(cc3CCn12)C#CCNc1ccccc1
Structure:
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