Reaction Details Report a problem with these data
Target
Melatonin receptor type 1A
Ligand
BDBM9019
Substrate
n/a
Meas. Tech.
ChEBML_105091
IC50
0.600000±n/a nM
Citation
Mattson, RJ; Catt, JD; Keavy, D; Sloan, CP; Epperson, J; Gao, Q; Hodges, DB; Iben, L; Mahle, CD; Ryan, E; Yocca, FD Indanyl piperazines as melatonergic MT2 selective agents. Bioorg Med Chem Lett 13:1199-202 (2003) [PubMed] Article
More Info.:
Target
Name:
Melatonin receptor type 1A
Synonyms:
MTNR1A | MTNR1A protein | MTR1A_HUMAN | Mel-1A-R | Mel1a melatonin receptor | Melatonin 1A | Melatonin receptor | Melatonin receptor 1A | Melatonin receptor type 1 (MT1) | Melatonin receptor type 1A
Type:
Enzyme
Mol. Mass.:
39392.94
Organism:
Homo sapiens (Human)
Description:
P48039
Residue:
350
Sequence:
MQGNGSALPNASQPVLRGDGARPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVADLVVAIYPYPLVLMSIFNNGWNLGYLHCQVSGFLMGLSVIGSIFNITGIAINRYCYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRQRVKPDRKPKLKPQDFRNFVTMFVVFVLFAICWAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNAIIYGLLNQNFRKEYRRIIVSLCTARVFFVDSSNDVADRVKWKPSPLMTNNNVVKVDSV