Reaction Details Report a problem with these data
Target
5'-3' exonuclease PLD3
Ligand
BDBM50572962
Substrate
n/a
Meas. Tech.
ChEMBL_2118712 (CHEMBL4827778)
IC50
39600±n/a nM
Citation
Shirey, RJ; Turner, LD; Lairson, LL; Janda, KD Modulators of immunoregulatory exonucleases PLD3 and PLD4 identified by high-throughput screen. Bioorg Med Chem Lett 49:0 (2021) [PubMed] Article
More Info.:
Target
Name:
5'-3' exonuclease PLD3
Synonyms:
3.1.16.1 | 5'-3' exonuclease PLD3 | Choline phosphatase 3 | HindIII K4L homolog | Hu-K4 | PLD 3 | PLD3 | PLD3_HUMAN | Phosphatidylcholine-hydrolyzing phospholipase D3 | Phospholipase D3
Type:
PROTEIN
Mol. Mass.:
54704.21
Organism:
Homo sapiens
Description:
ChEMBL_12540
Residue:
490
Sequence:
MKPKLMYQELKVPAEEPANELPMNEIEAWKAAEKKARWVLLVLILAVVGFGALMTQLFLWEYGDLHLFGPNQRPAPCYDPCEAVLVESIPEGLDFPNASTGNPSTSQAWLGLLAGAHSSLDIASFYWTLTNNDTHTQEPSAQQGEEVLRQLQTLAPKGVNVRIAVSKPSGPQPQADLQALLQSGAQVRMVDMQKLTHGVLHTKFWVVDQTHFYLGSANMDWRSLTQVKELGVVMYNCSCLARDLTKIFEAYWFLGQAGSSIPSTWPRFYDTRYNQETPMEICLNGTPALAYLASAPPPLCPSGRTPDLKALLNVVDNARSFIYVAVMNYLPTLEFSHPHRFWPAIDDGLRRATYERGVKVRLLISCWGHSEPSMRAFLLSLAALRDNHTHSDIQVKLFVVPADEAQARIPYARVNHNKYMVTERATYIGTSNWSGNYFTETAGTSLLVTQNGRGGLRSQLEAIFLRDWDSPYSHDLDTSADSVGNACRLL