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Target
Melatonin receptor type 1A
Ligand
BDBM50142203
Substrate
n/a
Meas. Tech.
ChEBML_104949
Ki
84±n/a nM
Citation
 Epperson, JR; Deskus, JA; Gentile, AJ; Iben, LG; Ryan, E; Sarbin, NS 4-Substituted anilides as selective melatonin MT2 receptor agonists. Bioorg Med Chem Lett 14:1023-6 (2004) [PubMed]  Article 
Target
Name:
Melatonin receptor type 1A
Synonyms:
MTNR1A | MTNR1A protein | MTR1A_HUMAN | Mel-1A-R | Mel1a melatonin receptor | Melatonin 1A | Melatonin receptor | Melatonin receptor 1A | Melatonin receptor type 1 (MT1) | Melatonin receptor type 1A
Type:
Enzyme
Mol. Mass.:
39392.94
Organism:
Homo sapiens (Human)
Description:
P48039
Residue:
350
Sequence:
MQGNGSALPNASQPVLRGDGARPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVADLVVAIYPYPLVLMSIFNNGWNLGYLHCQVSGFLMGLSVIGSIFNITGIAINRYCYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRQRVKPDRKPKLKPQDFRNFVTMFVVFVLFAICWAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNAIIYGLLNQNFRKEYRRIIVSLCTARVFFVDSSNDVADRVKWKPSPLMTNNNVVKVDSV
  
Inhibitor
Name:
BDBM50142203
Synonyms:
CHEMBL8094 | N-[4-(3-Methoxy-phenoxy)-phenyl]-acetamide
Type:
Small organic molecule
Emp. Form.:
C15H15NO3
Mol. Mass.:
257.2845
SMILES:
COc1cccc(Oc2ccc(NC(C)=O)cc2)c1
Structure:
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