Reaction Details Report a problem with these data
Target
Cell division protein FtsZ
Ligand
BDBM50581024
Substrate
n/a
Meas. Tech.
ChEMBL_2149614 (CHEMBL5034076)
Kd
1300±n/a nM
Citation
Huecas, S; Araújo-Bazán, L; Ruiz, FM; Ruiz-Ávila, LB; Martínez, RF; Escobar-Peńa, A; Artola, M; Vázquez-Villa, H; Martín-Fontecha, M; Fernández-Tornero, C; López-Rodríguez, ML; Andreu, JM Targeting the FtsZ Allosteric Binding Site with a Novel Fluorescence Polarization Screen, Cytological and Structural Approaches for Antibacterial Discovery. J Med Chem 64:5730-5745 (2021) [PubMed] Article
More Info.:
Target
Name:
Cell division protein FtsZ
Synonyms:
n/a
Type:
PROTEIN
Mol. Mass.:
40375.29
Organism:
Bacillus subtilis
Description:
ChEMBL_107642
Residue:
382
Sequence:
MLEFETNIDGLASIKVIGVGGGGNNAVNRMIENEVQGVEYIAVNTDAQALNLSKAEVKMQIGAKLTRGLGAGANPEVGKKAAEESKEQIEEALKGADMVFVTAGMGGGTGTGAAPVIAQIAKDLGALTVGVVTRPFTFEGRKRQLQAAGGISAMKEAVDTLIVIPNDRILEIVDKNTPMLEAFREADNVLRQGVQGISDLIATPGLINLDFADVKTIMSNKGSALMGIGIATGENRAAEAAKKAISSPLLEAAIDGAQGVLMNITGGTNLSLYEVQEAADIVASASDQDVNMIFGSVINENLKDEIVVTVIATGFIEQEKDVTKSQRPSLNQSIKTHNQSVPKREPKREEPQQQNTVSRHTSQPADDTLDIPTFLRNRNKRG