Reaction Details Report a problem with these data
Target
Adenosine receptor A2a
Ligand
BDBM50397728
Substrate
n/a
Meas. Tech.
ChEMBL_2157710 (CHEMBL5042370)
Ki
830±n/a nM
Citation
Suresh, RR; Gao, ZG; Salmaso, V; Chen, E; Campbell, RG; Poe, RB; Liston, TE; Jacobson, KA Selective A ACS Med Chem Lett 13:623-631 (2022) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A2a
Synonyms:
AA2AR_MOUSE | Adenosine A2a receptor | Adenosine receptor A2a | Adora2a
Type:
PROTEIN
Mol. Mass.:
44984.04
Organism:
Mus musculus
Description:
ChEMBL_479903
Residue:
410
Sequence:
MGSSVYIMVELAIAVLAILGNVLVCWAVWINSNLQNVTNFFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFFACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGMRAKGIIAICWVLSFAIGLTPMLGWNNCSQKDENSTKTCGEGRVTCLFEDVVPMNYMVYYNFFAFVLLPLLLMLAIYLRIFLAARRQLKQMESQPLPGERTRSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCSTCQHAPPWLMYLAIILSHSNSVVNPFIYAYRIREFRQTFRKIIRTHVLRRQEPFRAGGSSAWALAAHSTEGEQVSLRLNGHPLGVWANGSAPHSGRRPNGYTLGPGGGGSTQGSPGDVELLTQEHQEGQEHPGLGDHLAQGRVGTASWSSEFAPS