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Target
Phospholipase A2 group V
Ligand
BDBM50591713
Substrate
n/a
Meas. Tech.
ChEMBL_2201656 (CHEMBL5114364)
IC50
1530±n/a nM
Citation
 Jiang, X; Wu, K; Bai, R; Zhang, P; Zhang, Y Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities. Eur J Med Chem 229:0 (2022) [PubMed] 
Target
Name:
Phospholipase A2 group V
Synonyms:
PA2G5_HUMAN | PLA2G5 | Phospholipase A2 group V | Secretory phospholipase A2, group V (sPLA2-V)
Type:
Protein
Mol. Mass.:
15682.61
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
138
Sequence:
MKGLLPLAWFLACSVPAVQGGLLDLKSMIEKVTGKNALTNYGFYGCYCGWGGRGTPKDGTDWCCWAHDHCYGRLEEKGCNIRTQSYKYRFAWGVVTCEPGPFCHVNLCACDRKLVYCLKRNLRSYNPQYQYFPNILCS
  
Inhibitor
Name:
BDBM50591713
Synonyms:
CHEMBL5207115
Type:
Small organic molecule
Emp. Form.:
C17H10N4O5
Mol. Mass.:
350.2851
SMILES:
[O-][N+](=O)c1ccc(-c2ccc3n2c2ccccc2[nH]c3=O)c(c1)[N+]([O-])=O
Structure:
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