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Target
Aurora kinase B
Ligand
BDBM50594273
Substrate
n/a
Meas. Tech.
ChEMBL_2211677 (CHEMBL5124626)
IC50
960±n/a nM
Citation
Furqan, M; Fayyaz, A; Firdous, F; Raza, H; Bilal, A; Saleem, RSZ; Shahzad-Ul-Hussan, S; Wang, D; Youssef, FS; Al Musayeib, NM; Ashour, ML; Hussain, H; Faisal, A Identification and Characterization of Natural and Semisynthetic Quinones as Aurora Kinase Inhibitors. J Nat Prod 85:1503-1513 (2022) [PubMed]
More Info.:
Target
Name:
Aurora kinase B
Synonyms:
AIK2 | AIM-1 | AIM1 | AIRK2 | ARK2 | AURKB | AURKB_HUMAN | Aurora B kinase (aurB) | Aurora B-INCENP | Aurora kinase 2 | Aurora kinase B (AURKB) | Aurora-related kinase 2 | STK-1 | STK1 | STK12 | STK5 | Serine/threonine-protein kinase aurora B
Type:
Protein
Mol. Mass.:
39327.72
Organism:
Homo sapiens (Human)
Description:
Q96GD4
Residue:
344
Sequence:
MAQKENSYPWPYGRQTAPSGLSTLPQRVLRKEPVTPSALVLMSRSNVQPTAAPGQKVMENSSGTPDILTRHFTIDDFEIGRPLGKGKFGNVYLAREKKSHFIVALKVLFKSQIEKEGVEHQLRREIEIQAHLHHPNILRLYNYFYDRRRIYLILEYAPRGELYKELQKSCTFDEQRTATIMEELADALMYCHGKKVIHRDIKPENLLLGLKGELKIADFGWSVHAPSLRRKTMCGTLDYLPPEMIEGRMHNEKVDLWCIGVLCYELLVGNPPFESASHNETYRRIVKVDLKFPASVPMGAQDLISKLLRHNPSERLPLAQVSAHPWVRANSRRVLPPSALQSVA