Reaction Details Report a problem with these data
Target
Voltage-dependent L-type calcium channel subunit beta-2
Ligand
BDBM50101971
Substrate
n/a
Meas. Tech.
ChEMBL_2254454 (CHEMBL5168664)
IC50
30±n/a nM
Citation
More Info.:
Target
Name:
Voltage-dependent L-type calcium channel subunit beta-2
Synonyms:
CAB2 | CACB2_HUMAN | CACNB2 | CACNLB2 | Calcium channel voltage-dependent subunit beta 2 | L-type calcium channel alpha-1c/beta-2/alpha2delta-1 | Lambert-Eaton myasthenic syndrome antigen B | MYSB
Type:
PROTEIN
Mol. Mass.:
73595.87
Organism:
Homo sapiens
Description:
ChEMBL_117734
Residue:
660
Sequence:
MVQRDMSKSPPTAAAAVAQEIQMELLENVAPAGALGAAAQSYGKGARRKNRFKGSDGSTSSDTTSNSFVRQGSADSYTSRPSDSDVSLEEDREAVRREAERQAQAQLEKAKTKPVAFAVRTNVSYSAAHEDDVPVPGMAISFEAKDFLHVKEKFNNDWWIGRLVKEGCEIGFIPSPVKLENMRLQHEQRAKQGKFYSSKSGGNSSSSLGDIVPSSRKSTPPSSAIDIDATGLDAEENDIPANHRSPKPSANSVTSPHSKEKRMPFFKKTEHTPPYDVVPSMRPVVLVGPSLKGYEVTDMMQKALFDFLKHRFEGRISITRVTADISLAKRSVLNNPSKHAIIERSNTRSSLAEVQSEIERIFELARTLQLVVLDADTINHPAQLSKTSLAPIIVYVKISSPKVLQRLIKSRGKSQAKHLNVQMVAADKLAQCPPELFDVILDENQLEDACEHLADYLEAYWKATHPPSSSLPNPLLSRTLATSSLPLSPTLASNSQGSQGDQRTDRSAPIRSASQAEEEPSVEPVKKSQHRSSSSAPHHNHRSGTSRGLSRQETFDSETQESRDSAYVEPKEDYSHDHVDHYASHRDHNHRDETHGSSDHRHRESRHRSRDVDREQDHNECNKQRSRHKSKDRYCEKDGEVISKKRNEAGEWNRDVYIRQ