Reaction Details
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Target
Pyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial
Ligand
BDBM50615071
Substrate
n/a
Meas. Tech.
ChEMBL_2299604
IC50
8000±n/a nM
Citation
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More Info.:
Target
Name:
Pyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial
Synonyms:
1.2.4.1 | PDHA1 | PDHE1-A type I | Pyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial
Type:
PROTEIN
Mol. Mass.:
43128.05
Organism:
Sus scrofa
Description:
ChEMBL_116756
Residue:
389
Sequence:
GKMLAAVSRVLSGVAQKPASRVLVASRTFANDATFEIKKCDLHRLEEGPPVTTVLTREDGLKYYRMMQTVRRMELKADQLYKQKIIRGFCHLCDGQEACCVGLEAGINPTDHLITAYRAHGFTFTRGLSVREILAELTGRRGGCGKGKGGSMHMYAKNFYGGNGIVGAQVPLGAGIALACKYNGKDEVCLTLYGDGAANQGQIFEAYNMAALWKLPCVFICENNRYGMGTSVERAAASTDYYKRGDFIPGLRVDGMDILCVREATRFAAAYCRSGKGPILMELQTYRYHGHSMSDPGVSYRTREEIQEVRSKSDPIMLLKDRMVNSNLASVEELKEIDVEVRKEIEDAAQFATADPEPPLEELGYHIYCNDPPFEVRGANQWIKFKSIS