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Target
Carbonic anhydrase 2
Ligand
BDBM50210909
Substrate
n/a
Meas. Tech.
ChEMBL_444150 (CHEMBL893309)
Kd
141±n/a nM
Citation
 Dudutiene, V; Baranauskiene, L; Matulis, D Benzimidazo[1,2-c][1,2,3]thiadiazole-7-sulfonamides as inhibitors of carbonic anhydrase. Bioorg Med Chem Lett 17:3335-8 (2007) [PubMed]  Article 
Target
Name:
Carbonic anhydrase 2
Synonyms:
CA2 | CAH2_BOVIN | Carbonic anhydrase | Carbonic anhydrase 2 | Carbonic anhydrase II | Carbonic anhydrase II (CA II) | Carbonic anhydrase II (CA-II)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29115.93
Organism:
Bos taurus
Description:
n/a
Residue:
260
Sequence:
MSHHWGYGKHNGPEHWHKDFPIANGERQSPVDIDTKAVVQDPALKPLALVYGEATSRRMVNNGHSFNVEYDDSQDKAVLKDGPLTGTYRLVQFHFHWGSSDDQGSEHTVDRKKYAAELHLVHWNTKYGDFGTAAQQPDGLAVVGVFLKVGDANPALQKVLDALDSIKTKGKSTDFPNFDPGSLLPNVLDYWTYPGSLTTPPLLESVTWIVLKEPISVSSQQMLKFRTLNFNAEGEPELLMLANWRPAQPLKNRQVRGFPK
  
Inhibitor
Name:
BDBM50210909
Synonyms:
3-chlorobenzimidazo[1,2-c][1,2,3]thiadiazole-7-sulfonamide | CHEMBL394355
Type:
Small organic molecule
Emp. Form.:
C8H5ClN4O2S2
Mol. Mass.:
288.734
SMILES:
NS(=O)(=O)c1ccc2nc3C(Cl)=S=Nn3c2c1
Structure:
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