Reaction Details Report a problem with these data
Target
Deoxyhypusine synthase
Ligand
BDBM50216786
Substrate
n/a
Meas. Tech.
ChEMBL_437263 (CHEMBL906657)
Ki
100±n/a nM
Citation
Kaiser, A; Hammels, I; Gottwald, A; Nassar, M; Zaghloul, MS; Motaal, BA; Hauber, J; Hoerauf, A Modification of eukaryotic initiation factor 5A from Plasmodium vivax by a truncated deoxyhypusine synthase from Plasmodium falciparum: An enzyme with dual enzymatic properties. Bioorg Med Chem 15:6200-7 (2007) [PubMed] Article
More Info.:
Target
Name:
Deoxyhypusine synthase
Synonyms:
n/a
Type:
PROTEIN
Mol. Mass.:
57187.86
Organism:
Plasmodium falciparum
Description:
ChEMBL_437263
Residue:
496
Sequence:
MVDHVSFIEVNKIRSDDECDADSHNEGDNIEDAKASVFVKSSLIPEKTDVVKGLNFDKEVDLHEFINNYKYMGFQATNLGISIDEINKMIYYKYKDENIKSEPNNENNLNCNNVSEDLNKDQENHLYHYEKKKKSCIIWLSFTSNMISSGLREIFVYLAKNKFIDVVVTTAGGIEEDIIKCFSNTYIGDFNLNGKKLRKKGWNRIGNLIVPNDNYCKFEDWLQPILNKMLHEQNEKNEQMFLKKLEKRKKKYNNNKNKNDNNNDNDNVWGNEKNDQNENQYNQGQESFKKDSNIYTNDVSNKKNHINNYINNYDSDSDDQCDMYYLSPSEFINTLGKEINDESSLIYWCYKNDIPIFCPGLTDGSLGDNLFLHNYGKKIKNNLILDIVKDIKKINSLAMNCEKSGIIILGGGLPKHHVCNANLMRNGADFAVYVNTASEYDGSDSGANTTEALSWGKIKYGQTNNHVKVFGDATILFPLMVLNSFYLYDQKRKKDM