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Target
Galectin-1
Ligand
BDBM50243734
Substrate
n/a
Meas. Tech.
ChEMBL_491861 (CHEMBL946198)
Kd
4400000±n/a nM
Citation
 Oberg, CT; Blanchard, H; Leffler, H; Nilsson, UJ Protein subtype-targeting through ligand epimerization: talose-selectivity of galectin-4 and galectin-8. Bioorg Med Chem Lett 18:3691-4 (2008) [PubMed]  Article 
Target
Name:
Galectin-1
Synonyms:
14 kDa lectin | Galaptin | HPL | LEG1_HUMAN | LGALS1 | Lactose-binding lectin 1 | Lectin galactoside-binding soluble 1 | Putative MAPK-activating protein PM12
Type:
beta galactoside-binding protein
Mol. Mass.:
14713.53
Organism:
Homo sapiens (Human)
Description:
P09382
Residue:
135
Sequence:
MACGLVASNLNLKPGECLRVRGEVAPDAKSFVLNLGKDSNNLCLHFNPRFNAHGDANTIVCNSKDGGAWGTEQREAVFPFQPGSVAEVCITFDQANLTVKLPDGYEFKFPNRLNLEAINYMAADGDFKIKCVAFD
  
Inhibitor
Name:
BDBM50243734
Synonyms:
CHEMBL479534 | triethylazanium (2R,3S,4S,5S,6R)-5-hydroxy-6-(hydroxymethyl)-2-methoxy-4-[(4-methylphenyl)carbonyloxy]oxan-3-yl (4-methylphenyl)methyl phosphate
Type:
Small organic molecule
Emp. Form.:
C23H28O10P
Mol. Mass.:
495.4367
SMILES:
CO[C@@H]1O[C@H](CO)[C@H](O)[C@H](OC(=O)c2ccc(C)cc2)[C@@H]1OP([O-])(=O)OCc1ccc(C)cc1 |r|
Structure:
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