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Target
Trace amine-associated receptor 1
Ligand
BDBM50022723
Substrate
n/a
Meas. Tech.
ChEMBL_489239 (CHEMBL989986)
EC50
935±n/a nM
Citation
 Lewin, AH; Navarro, HA; Mascarella, SW Structure-activity correlations for beta-phenethylamines at human trace amine receptor 1. Bioorg Med Chem 16:7415-23 (2008) [PubMed]  Article 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TAAR1_HUMAN | TAAR1 | TA1 | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:
PROTEIN
Mol. Mass.:
39107.47
Organism:
Human
Description:
ChEMBL_792734
Residue:
339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNWLIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISIDRYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRGGCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNGISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFNPMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
  
Inhibitor
Name:
BDBM50022723
Synonyms:
(2S)-1-phenylpropan-2-amine | (S)-amphetamine | (+)-(S)-amphetamine | (+)-alpha-methylphenethylamine | (+)-alpha-methylphenylethylamine | (S)-(+)-amphetamine | (S)-(+)-beta-phenylisopropylamine | (S)-1-phenyl-2-aminopropane | (S)-1-phenyl-2-propylamine | (S)-alpha-methylbenzeneethanamine | (alphaS)-alpha-methylbenzeneethanamine | Dextroamphetamine | d-amphetamine | dexamphetamine | CHEMBL612
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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