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Target
Protein kinase domain-containing protein
Ligand
BDBM50264944
Substrate
n/a
Meas. Tech.
ChEMBL_496798 (CHEMBL1008811)
IC50
7400±n/a nM
Citation
Bouloc, N; Large, JM; Smiljanic, E; Whalley, D; Ansell, KH; Edlin, CD; Bryans, JS Synthesis and in vitro evaluation of imidazopyridazines as novel inhibitors of the malarial kinase PfPK7. Bioorg Med Chem Lett 18:5294-8 (2008) [PubMed] Article
More Info.:
Target
Name:
Protein kinase domain-containing protein
Synonyms:
Putative uncharacterized protein pk7
Type:
PROTEIN
Mol. Mass.:
37967.83
Organism:
Plasmodium falciparum
Description:
ChEMBL_496798
Residue:
320
Sequence:
MKDILSNYSNLIYLNKYVKEKDKYINDYRIIRTLNQGKFNKIILCEKDNKFYALKKYEKSLLEKKRDFTKSNNDKISIKSKYDDFKNELQIITDIKNEYCLTCEGIITNYDEVYIIYEYMENDSILKFDEYFFVLDKNYTCFIPIQVIKCIIKSVLNSFSYIHNEKNICHRDVKPSNILMDKNGRVKLSDFGESEYMVDKKIKGSRGTYEFMPPEFFSNESSYNGAKVDIWSLGICLYVMFYNVVPFSLKISLVELFNNIRTKNIEYPLDRNHFLYPLTNKKSTCSNNFLSNEDIDFLKLFLRKNPAERITSEDALVTAK