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Target
D(2) dopamine receptor
Ligand
BDBM50283337
Substrate
n/a
Meas. Tech.
ChEBML_61122
Ki
>10000±n/a nM
Citation
 Christos, TE; Cain, GA; Johnson, AL; Schmidt, WK; Tam, SW Novel ether derivatives of alkyl piperidines as potential sigma / 5HT2 antipsychotic agents Bioorg Med Chem Lett 4:2347-2352 (1994)    Article 
Target
Name:
D(2) dopamine receptor
Synonyms:
D(2) dopamine receptor | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2 | DRD2_HUMAN | Dopamine D2 receptor | Dopamine D2 receptor (D2) | Dopamine D2 receptor (D2R) | Dopamine D2A | Dopamine2-like | d2
Type:
Cell-surface receptors
Mol. Mass.:
50647.10
Organism:
Homo sapiens (Human)
Description:
P14416
Residue:
443
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSDGKADRPHYNYYATLLTLLIAVIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMISIVWVLSFTISCPLLFGLNNADQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTKRSSRAFRAHLRAPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSTPDSPAKPEKNGHAKDHPKIAKIFEIQTMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFLKILHC
  
Inhibitor
Name:
BDBM50283337
Synonyms:
1-Benzyl-4-((1E,3E)-4-phenyl-buta-1,3-dienyloxymethyl)-piperidine | CHEMBL80784
Type:
Small organic molecule
Emp. Form.:
C23H27NO
Mol. Mass.:
333.4666
SMILES:
C(O\C=C\C=C\c1ccccc1)C1CCN(Cc2ccccc2)CC1
Structure:
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