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Target
Mu-type opioid receptor
Ligand
BDBM50450285
Substrate
n/a
Meas. Tech.
ChEBML_136093
IC50
5.1±n/a nM
Citation
 Kudzma, LV; Evans, SM; Turnbull, SP; Severnak, SA; Ezell, EF Octahydro-1,2,3,4,4a,5,11,11a-pyrido[3,4-c][1,5]benzoxazepines: conformationally restricted fentanyl analogs Bioorg Med Chem Lett 5:1177-1182 (1995)    Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50450285
Synonyms:
CHEMBL2079638
Type:
Small organic molecule
Emp. Form.:
C23H28N2O2
Mol. Mass.:
364.4806
SMILES:
[H][C@@]12CN(CCc3ccccc3)CCC1N(C(=O)CC)c1ccccc1OC2 |r|
Structure:
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