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Target
D(2) dopamine receptor
Ligand
BDBM50054398
Substrate
n/a
Meas. Tech.
ChEBML_62406
Ki
>10000±n/a nM
Citation
 López-Rodríguez, ML; Morcillo, M; Rosado, M; Benhamu, B; Sanz, AM 2-[4-(o-methoxyphenyl)piperazin-1-ylmethyl]-1,3-dioxoperhydroimidazo[1,5-a]pyridine as a new selective 5-HT1A receptor ligand Bioorg Med Chem Lett 6:689-694 (1996)    Article 
Target
Name:
D(2) dopamine receptor
Synonyms:
DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
50931.60
Organism:
Rattus norvegicus (rat)
Description:
P61169
Residue:
444
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSEGKADRPHYNYYAMLLTLLIFIIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFMKILHC
  
Inhibitor
Name:
BDBM50054398
Synonyms:
2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-tetrahydro-imidazo[1,5-a]pyridine-1,3-dione | CHEMBL295168
Type:
Small organic molecule
Emp. Form.:
C19H26N4O3
Mol. Mass.:
358.4347
SMILES:
COc1ccccc1N1CCN(Cn2c(O)c3CCCCn3c2=O)CC1
Structure:
Search PDB for entries with ligand similarity: