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Target
Prostatic acid phosphatase
Ligand
BDBM50288656
Substrate
n/a
Meas. Tech.
ChEBML_158625
IC50
14000±n/a nM
Citation
 Frechette, RF; Ackerman, C; Beers, S; Look, R; Moore, J Novel hydroxyphosphonate inhibitors of CD-45 tyrosine phosphatase Bioorg Med Chem Lett 7:2169-2172 (1997)    Article 
Target
Name:
Prostatic acid phosphatase
Synonyms:
ACP3 | ACPP | PPAP_HUMAN | Prostatic acid phosphatase
Type:
PROTEIN
Mol. Mass.:
44563.07
Organism:
Homo sapiens (Human)
Description:
ChEMBL_158625
Residue:
386
Sequence:
MRAAPLLLARAASLSLGFLFLLFFWLDRSVLAKELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRFQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMTTNSHQGTEDSTD
  
Inhibitor
Name:
BDBM50288656
Synonyms:
(Phenyl-m-tolyl-methyl)-phosphonic acid | CHEMBL71259
Type:
Small organic molecule
Emp. Form.:
C14H15O3P
Mol. Mass.:
262.2409
SMILES:
Cc1cccc(c1)C(c1ccccc1)P(O)(O)=O
Structure:
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