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Target
D(1A) dopamine receptor
Ligand
BDBM50298910
Substrate
n/a
Meas. Tech.
ChEMBL_588133 (CHEMBL1044859)
Ki
4100±n/a nM
Citation
 Loaiza, PR; Löber, S; Hübner, H; Gmeiner, P Parallel synthesis of potent dopaminergic N-phenyltriazole carboxamides applying a novel click chemistry based phenol linker. Bioorg Med Chem 17:5482-7 (2009) [PubMed]  Article 
Target
Name:
D(1A) dopamine receptor
Synonyms:
DRD1 | DRD1_PIG | Dopamine D1 receptor
Type:
PROTEIN
Mol. Mass.:
49269.92
Organism:
Sus scrofa
Description:
ChEMBL_1460140
Residue:
446
Sequence:
MRTLNTSTMDGTGLVVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNVTSLGKTTHNCDSSLSRTYAISSSLISFYIPVAIMIVTYTRIYRIAQKQIRRISALERAAVHAKNCQTTAGNGNPAECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCGSGETKPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPTSTNAIETVSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIASPLEKLSPALSVILDYDTDVSLEKIQPITQNGQHPT
  
Inhibitor
Name:
BDBM50298910
Synonyms:
CHEMBL573791 | N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1-(4-nitrophenyl)-1H-1,2,3-triazole-4-carboxamide
Type:
Small organic molecule
Emp. Form.:
C22H25N7O4
Mol. Mass.:
451.4784
SMILES:
COc1ccccc1N1CCN(CCNC(=O)c2cn(nn2)-c2ccc(cc2)[N+]([O-])=O)CC1
Structure:
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