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Target
D(1A) dopamine receptor
Ligand
BDBM50298914
Substrate
n/a
Meas. Tech.
ChEMBL_588133 (CHEMBL1044859)
Ki
140±n/a nM
Citation
 Loaiza, PR; Löber, S; Hübner, H; Gmeiner, P Parallel synthesis of potent dopaminergic N-phenyltriazole carboxamides applying a novel click chemistry based phenol linker. Bioorg Med Chem 17:5482-7 (2009) [PubMed]  Article 
Target
Name:
D(1A) dopamine receptor
Synonyms:
DRD1 | DRD1_PIG | Dopamine D1 receptor
Type:
PROTEIN
Mol. Mass.:
49269.92
Organism:
Sus scrofa
Description:
ChEMBL_1460140
Residue:
446
Sequence:
MRTLNTSTMDGTGLVVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNVTSLGKTTHNCDSSLSRTYAISSSLISFYIPVAIMIVTYTRIYRIAQKQIRRISALERAAVHAKNCQTTAGNGNPAECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCGSGETKPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPTSTNAIETVSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIASPLEKLSPALSVILDYDTDVSLEKIQPITQNGQHPT
  
Inhibitor
Name:
BDBM50298914
Synonyms:
CHEMBL572867 | N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(1-(4-methoxyphenyl)-1H-1,2,3-triazol-4-yl)butanamide
Type:
Small organic molecule
Emp. Form.:
C27H34Cl2N6O2
Mol. Mass.:
545.504
SMILES:
COc1ccc(cc1)-n1cc(CCCC(=O)NCCCCN2CCN(CC2)c2cccc(Cl)c2Cl)nn1
Structure:
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