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Target
Transthyretin
Ligand
BDBM60927
Substrate
n/a
Meas. Tech.
ChEMBL_607502 (CHEMBL1070778)
Kd
4800±n/a nM
Citation
Lima, LM; Silva, Vde A; Palmieri, Lde C; Oliveira, MC; Foguel, D; Polikarpov, I Identification of a novel ligand binding motif in the transthyretin channel. Bioorg Med Chem 18:100-10 (2010) [PubMed] Article
More Info.:
Target
Name:
Transthyretin
Synonyms:
ATTR | PALB | Prealbumin | TBPA | TTHY_HUMAN | TTR | Transthyretin (TTR)
Type:
Enzyme
Mol. Mass.:
15884.31
Organism:
Human
Description:
P02766
Residue:
147
Sequence:
MASHRLLLLCLAGLVFVSEAGPTGTGESKCPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNPKE