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Target
Mu-type opioid receptor
Ligand
BDBM50320088
Substrate
n/a
Meas. Tech.
ChEMBL_635249 (CHEMBL1118189)
Ki
24.7±n/a nM
Citation
 Nagase, H; Imaide, S; Tomatsu, M; Nemoto, T; Nakajima, M; Nakao, K; Mochizuki, H; Fujii, H Investigation of Beckett-Casy model 2: synthesis of novel 15-16 nornaltrexone derivatives and their pharmacology. Bioorg Med Chem Lett 20:3726-9 (2010) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50320088
Synonyms:
(2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-dihydroxy-2,2a,2a1,3,4,5a-hexahydrophenanthro[4,5-bcd]furan-5(1H)-one | CHEMBL1082639
Type:
Small organic molecule
Emp. Form.:
C18H21NO4
Mol. Mass.:
315.3636
SMILES:
Oc1ccc2C[C@@H](NCC3CC3)[C@]3(O)CCC(=O)[C@@H]4Oc1c2[C@H]34 |r|
Structure:
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