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Target
Mu-type opioid receptor
Ligand
BDBM50357429
Substrate
n/a
Meas. Tech.
ChEMBL_788480 (CHEMBL1918283)
Ki
92±n/a nM
Citation
 Rossi, D; Pedrali, A; Urbano, M; Gaggeri, R; Serra, M; Fernández, L; Fernández, M; Caballero, J; Ronsisvalle, S; Prezzavento, O; Schepmann, D; Wuensch, B; Peviani, M; Curti, D; Azzolina, O; Collina, S Identification of a potent and selectives¿? receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells. Bioorg Med Chem 19:6210-24 (2011) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50357429
Synonyms:
CHEMBL1917702
Type:
Small organic molecule
Emp. Form.:
C19H23NO
Mol. Mass.:
281.392
SMILES:
COc1ccc(cc1)C(\C)=C\CN(C)Cc1ccccc1
Structure:
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