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Target
D(2) dopamine receptor
Ligand
BDBM50029344
Substrate
n/a
Meas. Tech.
ChEMBL_63059 (CHEMBL673626)
Ki
3570±n/a nM
Citation
 Shah, JH; Izenwasser, S; Geter-Douglass, B; Witkin, JM; Newman, AH (+/-)-(N-alkylamino)benzazepine analogs: novel dopamine D1 receptor antagonists. J Med Chem 38:4284-93 (1995) [PubMed]  Article 
Target
Name:
D(2) dopamine receptor
Synonyms:
DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
50931.60
Organism:
Rattus norvegicus (rat)
Description:
P61169
Residue:
444
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSEGKADRPHYNYYAMLLTLLIFIIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFMKILHC
  
Inhibitor
Name:
BDBM50029344
Synonyms:
8-Chloro-3-(6-methylamino-hexyl)-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol | CHEMBL108480
Type:
Small organic molecule
Emp. Form.:
C23H31ClN2O
Mol. Mass.:
386.958
SMILES:
CNCCCCCCN1CCc2cc(Cl)c(O)cc2C(C1)c1ccccc1
Structure:
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