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Target
Somatostatin receptor type 5
Ligand
BDBM50169478
Substrate
n/a
Meas. Tech.
ChEMBL_302433 (CHEMBL827131)
Ki
56±n/a nM
Citation
 Contour-Galcéra, MO; Sidhu, A; Plas, P; Roubert, P 3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists. Bioorg Med Chem Lett 15:3555-9 (2005) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5)
Type:
Enzyme
Mol. Mass.:
39218.02
Organism:
Homo sapiens (Human)
Description:
P35346
Residue:
364
Sequence:
MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTLVIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDGVNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADVQEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRRRSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCANPVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQTSKL
  
Inhibitor
Name:
BDBM50169478
Synonyms:
4-{3-[2-(1H-Indol-3-yl)-ethylsulfanyl]-5-quinoxalin-2-yl-[1,2,4]triazol-4-yl}-butylamine | CHEMBL188402
Type:
Small organic molecule
Emp. Form.:
C24H25N7S
Mol. Mass.:
443.567
SMILES:
NCCCCn1c(SCCc2c[nH]c3ccccc23)nnc1-c1cnc2ccccc2n1
Structure:
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