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Target
Mu-type opioid receptor
Ligand
BDBM50194242
Substrate
n/a
Meas. Tech.
ChEMBL_392093 (CHEMBL869901)
IC50
53.9±n/a nM
Citation
 Balboni, G; Onnis, V; Congiu, C; Zotti, M; Sasaki, Y; Ambo, A; Bryant, SD; Jinsmaa, Y; Lazarus, LH; Trapella, C; Salvadori, S Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore. J Med Chem 49:5610-7 (2006) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50194242
Synonyms:
CHEMBL378082 | H-Dmt-Tic-NH-CH[(CH2)4-NH-Ac]-Bid
Type:
Small organic molecule
Emp. Form.:
C35H42N6O4
Mol. Mass.:
610.7458
SMILES:
CC(=O)NCCCCC(NC(=O)C1Cc2ccccc2CN1C(=O)C(N)Cc1c(C)cc(O)cc1C)c1nc2ccccc2[nH]1
Structure:
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