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Target
Amine oxidase [flavin-containing] A
Ligand
BDBM50217273
Substrate
n/a
Meas. Tech.
ChEMBL_440608 (CHEMBL889702)
IC50
>150000±n/a nM
Citation
 Hwang, JH; Hong, SS; Han, XH; Hwang, JS; Lee, D; Lee, H; Yun, YP; Kim, Y; Ro, JS; Hwang, BY Prenylated xanthones from the root bark of Cudrania tricuspidata. J Nat Prod 70:1207-9 (2007) [PubMed]  Article 
Target
Name:
Amine oxidase [flavin-containing] A
Synonyms:
AOFA_MOUSE | Amine oxidase [flavin-containing] A | MAO-A | Maoa | Monoamine oxidase | Monoamine oxidase A | Monoamine oxidase type A
Type:
PROTEIN
Mol. Mass.:
59608.24
Organism:
Mus musculus
Description:
ChEMBL_122776
Residue:
526
Sequence:
MTDLEKPSITGHMFDVVVIGGGISGLAAAKLLSEYKINVLVLEARDRVGGRTYTVRNEHVKWVDVGGAYVGPTQNRILRLSKELGIETYKVNVNERLVQYVKGKTYPFRGAFPPVWNPLAYLDYNNLWRTMDDMGKEIPVDAPWQARHAEEWDKITMKDLIDKICWTKTAREFAYLFVNINVTSEPHEVSALWFLWYVRQCGGTSRIFSVTNGGQERKFVGGSGQISEQIMVLLGDKVKLSSPVTYIDQTDDNIIIETLNHEHYECKYVISAIPPVLTAKIHFKPELPPERNQLIQRLPMGAVIKCMVYYKEAFWKKKDYCGCMIIEDEEAPISITLDDTKPDGSMPAIMGFILARKAERLAKLHKDIRKRKICELYAKVLGSQEALSPVHYEEKNWCEEQYSGGCYTAYFPPGIMTLYGRVIRQPVGRIYFAGTETATQWSGYMEGAVEAGERAAREVLNALGKVAKKDIWVQEPESKDVPALEITHTFLERNLPSVPGLLKITGFSTSVALLCFVLYKFKQPQS
  
Inhibitor
Name:
BDBM50217273
Synonyms:
CHEMBL390040 | isocudraxanthone K
Type:
Small organic molecule
Emp. Form.:
C23H22O6
Mol. Mass.:
394.4172
SMILES:
CC(C)(C=C)c1c(O)cc2oc3c4C=CC(C)(C)Oc4c(O)cc3c(=O)c2c1O |c:13|
Structure:
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