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Target
Mu-type opioid receptor
Ligand
BDBM50347178
Substrate
n/a
Meas. Tech.
ChEMBL_753740 (CHEMBL1799577)
Ki
0.16±n/a nM
Citation
 Yamamoto, N; Fujii, H; Nemoto, T; Nakajima, R; Momen, S; Izumimoto, N; Hasebe, K; Mochizuki, H; Nagase, H Synthesis of new opioid derivatives with a propellane skeleton and their pharmacology: part 1. Bioorg Med Chem Lett 21:4104-7 (2011) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50347178
Synonyms:
CHEMBL1797688
Type:
Small organic molecule
Emp. Form.:
C21H25NO4
Mol. Mass.:
355.4275
SMILES:
Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45C(Oc1c24)C1(O)CC[C@@]35OC1 |r|
Structure:
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