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Target
Prostaglandin E2 receptor EP2 subtype
Ligand
BDBM50385133
Substrate
n/a
Meas. Tech.
ChEMBL_822927 (CHEMBL2038098)
Ki
15±n/a nM
Citation
 Kambe, T; Maruyama, T; Nakai, Y; Oida, H; Maruyama, T; Abe, N; Nishiura, A; Nakai, H; Toda, M Synthesis and evaluation of¿-lactam analogs of PGE2 as EP4 and EP2/EP4 agonists. Bioorg Med Chem 20:3502-22 (2012) [PubMed]  Article 
Target
Name:
Prostaglandin E2 receptor EP2 subtype
Synonyms:
Prostaglandin E2 | Prostaglandin E2 receptor EP2 subtype | PGE receptor, EP2 subtype | PE2R2_MOUSE | Ptger2 | Ptgerep2 | Prostanoid EP2 receptor
Type:
G-protein coupled receptor
Mol. Mass.:
40495.26
Organism:
Mouse
Description:
n/a
Residue:
362
Sequence:
MDNFLNDSKLMEDCKSRQWLLSGESPAISSVMFSAGVLGNLIALALLARRWRGDTGCSAGSRTSISLFHVLVTELVLTDLLGTCLISPVVLASYSRNQTLVALAPESHACTYFAFTMTFFSLATMLMLFAMALERYLSIGYPYFYRRHLSRRGGLAVLPVIYGASLLFCSLPLLNYGEYVQYCPGTWCFIRHGRTAYLQLYATMLLLLIVAVLACNISVILNLIRMHRRSRRSRCGLSGSSLRGPGSRRRGERTSMAEETDHLILLAIMTITFAICSLPFTIFAYMDETSSLKEKWDLRALRFLSVNSIIDPWVFAILRPPVLRLMRSVLCCRTSLRTQEAQQTSCSTQSSASKQTDLCGQL
  
Inhibitor
Name:
BDBM50385133
Synonyms:
CHEMBL2036324
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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