Reaction Details Report a problem with these data
Target
Free fatty acid receptor 1
Ligand
BDBM50339456
Substrate
n/a
Meas. Tech.
ChEMBL_830235 (CHEMBL2060786)
EC50
549.54±n/a nM
Citation
 Shimpukade, B; Hudson, BD; Hovgaard, CK; Milligan, G; Ulven, T Discovery of a potent and selective GPR120 agonist. J Med Chem 55:4511-5 (2012) [PubMed]  Article 
Target
Name:
Free fatty acid receptor 1
Synonyms:
FFAR1 | FFAR1_HUMAN | G-protein Coupled Receptor 40 | GPR40
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
31473.32
Organism:
Homo sapiens (Human)
Description:
O14842
Residue:
300
Sequence:
MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSLVYALNLGCSDLLLTVSLPLKAVEALASGAWPLPASLCPVFAVAHFFPLYAGGGFLAALSAGRYLGAAFPLGYQAFRRPCYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAGPARFSLSLLLFFLPLAITAFCYVGCLRALARSGLTHRRKLRAAWVAGGALLTLLLCVGPYNASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLGRGPGLKTVCAARTQGGKSQK
  
Inhibitor
Name:
BDBM50339456
Synonyms:
Benzyloxyphenylpropanoic acid | CHEMBL1688452
Type:
Small organic molecule
Emp. Form.:
C16H16O3
Mol. Mass.:
256.2964
SMILES:
OC(=O)CCc1ccc(OCc2ccccc2)cc1
Structure:
Search PDB for entries with ligand similarity: