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Target
Solute carrier family 22 member 1
Ligand
BDBM50149890
Substrate
n/a
Meas. Tech.
ChEMBL_835933 (CHEMBL2077071)
IC50
540±n/a nM
Citation
 Kakehi, M; Koyabu, N; Nakamura, T; Uchiumi, T; Kuwano, M; Ohtani, H; Sawada, Y Functional characterization of mouse cation transporter mOCT2 compared with mOCT1. Biochem Biophys Res Commun 296:644-50 (2002) [PubMed]  Article 
Target
Name:
Solute carrier family 22 member 1
Synonyms:
Lx1 | Oct1 | Organic cation transporter 1 | S22A1_MOUSE | Slc22a1 | mOCT1
Type:
PROTEIN
Mol. Mass.:
61521.43
Organism:
Mus musculus
Description:
ChEMBL_1279071
Residue:
556
Sequence:
MPTVDDVLEHVGEFGWFQKQAFLLLCLISASLAPIYVGIVFLGFTPDHHCRSPGVAELSQRCGWSPAEELNYTVPGLGSAGEASFLSQCMKYEVDWNQSTLDCVDPLSSLAANRSHLPLSPCEHGWVYDTPGSSIVTEFNLVCGDAWKVDLFQSCVNLGFFLGSLVVGYIADRFGRKLCLLVTTLVTSLSGVLTAVAPDYTSMLLFRLLQGMVSKGSWVSGYTLITEFVGSGYRRTTAILYQVAFTVGLVGLAGVAYAIPDWRWLQLAVSLPTFLFLLYYWFVPESPRWLLSQKRTTQAVRIMEQIAQKNRKVPPADLKMMCLEEDASERRSPSFADLFRTPSLRKHTLILMYLWFSCAVLYQGLIMHVGATGANLYLDFFYSSLVEFPAAFIILVTIDRIGRIYPIAASNLVAGAACLLMIFIPHELHWLNVTLACLGRMGATIVLQMVCLVNAELYPTFIRNLGMMVCSALCDLGGIFTPFMVFRLMEVWQALPLILFGVLGLSAGAVTLLLPETKGVALPETIEEAENLGRRKSKAKENTIYLQVQTGKSPHT
  
Inhibitor
Name:
BDBM50149890
Synonyms:
CHEMBL9324 | tetraethylammonium
Type:
Small organic molecule
Emp. Form.:
C8H20N
Mol. Mass.:
130.2506
SMILES:
CC[N+](CC)(CC)CC
Structure:
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