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Target
G-protein coupled receptor 55
Ligand
BDBM50398241
Substrate
n/a
Meas. Tech.
ChEMBL_963381 (CHEMBL2388878)
IC50
3990±n/a nM
Citation
 Rempel, V; Volz, N; Gläser, F; Nieger, M; Bräse, S; Müller, CE Antagonists for the orphan G-protein-coupled receptor GPR55 based on a coumarin scaffold. J Med Chem 56:4798-810 (2013) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 55
Synonyms:
G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN
Type:
PROTEIN
Mol. Mass.:
36649.72
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1292265
Residue:
319
Sequence:
MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATSIYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRFLAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAKVFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFLPVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIRAHRPSRVQLVLQDTTISRG
  
Inhibitor
Name:
BDBM50398241
Synonyms:
CHEMBL2181551
Type:
Small organic molecule
Emp. Form.:
C18H15BrO4
Mol. Mass.:
375.213
SMILES:
COc1cccc(Cc2cc3c(OC)cc(Br)cc3oc2=O)c1
Structure:
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