Reaction Details Report a problem with these data
Target
Thymidine kinase, cytosolic
Ligand
BDBM50000975
Substrate
n/a
Meas. Tech.
ChEMBL_1333876 (CHEMBL3231765)
Ki
4400000±n/a nM
Citation
Hampton, A; Kappler, F; Chawla, RR Design of species- or isozyme-specific enzyme inhibitors. 1. Effect of thymidine substituents on affinity for the thymidine site of hamster cytoplasmic thymidine kinase. J Med Chem 22:621-31 (1979) [PubMed] Article
More Info.:
Target
Name:
Thymidine kinase, cytosolic
Synonyms:
KITH_CRIGR | TK1
Type:
PROTEIN
Mol. Mass.:
25628.94
Organism:
Cricetulus griseus
Description:
ChEMBL_108265
Residue:
234
Sequence:
MNYINLPTVLPGSPSKTRGQIQVILGPMFSGKSTELMRRVRRFQIAQNKCLVIKYAKDTRYSSSFSTHDRNTMDALPACLLRDVAQEALGAAVIGIDEGQFFPDIVEFCEVMANAGKTVIVAALDGTFQRKAFGSILNLVPLAESVVKLTAVCMECFREAAYTKRLGLEKEVEVIGGADKYHSVCRVCYFKKSSVQPAGPDNKENCPVLGQPGEASAVRKLFAPQQVLQHNSTN