Reaction Details Report a problem with these data
Target
G-protein coupled receptor 52
Ligand
BDBM50022156
Substrate
n/a
Meas. Tech.
ChEMBL_1367592
EC50
35±n/a nM
Citation
Setoh, M; Ishii, N; Kono, M; Miyanohana, Y; Shiraishi, E; Harasawa, T; Ota, H; Odani, T; Kanzaki, N; Aoyama, K; Hamada, T; Kori, M Discovery of the first potent and orally available agonist of the orphan G-protein-coupled receptor 52. J Med Chem 57:5226-37 (2014) [PubMed] Article
More Info.:
Target
Name:
G-protein coupled receptor 52
Synonyms:
GPR52 | GPR52_HUMAN | Probable G-protein coupled receptor 52
Type:
PROTEIN
Mol. Mass.:
41366.15
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108391
Residue:
361
Sequence:
MNESRWTEWRILNMSSGIVNVSERHSCPLGFGHYSVVDVCIFETVVIVLLTFLIIAGNLTVIFVFHCAPLLHHYTTSYFIQTMAYADLFVGVSCLVPTLSLLHYSTGVHESLTCQVFGYIISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIILIWIYSCLIFLPSFFGWGKPGYHGDIFEWCATSWLTSAYFTGFIVCLLYAPAAFVVCFTYFHIFKICRQHTKEINDRRARFPSHEVDSSRETGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSFLTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCMCVKDQEAQEPKPRKRANSCSI