Reaction Details Report a problem with these data
Target
40S ribosomal protein S27
Ligand
BDBM50048362
Substrate
n/a
Meas. Tech.
ChEMBL_1446775 (CHEMBL3381090)
IC50
>10000±n/a nM
Citation
Casale, E; Amboldi, N; Brasca, MG; Caronni, D; Colombo, N; Dalvit, C; Felder, ER; Fogliatto, G; Galvani, A; Isacchi, A; Polucci, P; Riceputi, L; Sola, F; Visco, C; Zuccotto, F; Casuscelli, F Fragment-based hit discovery and structure-based optimization of aminotriazoloquinazolines as novel Hsp90 inhibitors. Bioorg Med Chem 22:4135-50 (2014) [PubMed] Article
More Info.:
Target
Name:
40S ribosomal protein S27
Synonyms:
MPS-1 | MPS1 | Metallopan-stimulin 1 | RPS27 | RS27_HUMAN
Type:
PROTEIN
Mol. Mass.:
9472.13
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1446775
Residue:
84
Sequence:
MPLAKDLLHPSPEEEKRKHKKKRLVQSPNSYFMDVKCPGCYKITTVFSHAQTVVLCVGCSTVLCQPTGGKARLTEGCSFRRKQH