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Target
Inhibitor of growth protein 2
Ligand
BDBM92788
Substrate
n/a
Meas. Tech.
ChEMBL_1566080 (CHEMBL3791708)
IC50
105000±n/a nM
Citation
 McAllister, TE; England, KS; Hopkinson, RJ; Brennan, PE; Kawamura, A; Schofield, CJ Recent Progress in Histone Demethylase Inhibitors. J Med Chem 59:1308-29 (2016) [PubMed]  Article 
Target
Name:
Inhibitor of growth protein 2
Synonyms:
ING1L | ING1Lp | ING2 | ING2_HUMAN | Inhibitor of growth 1-like protein | Inhibitor of growth protein 2 | p32 | p33ING2
Type:
PROTEIN
Mol. Mass.:
32812.71
Organism:
Homo sapiens (Human)
Description:
ChEMBL_116766
Residue:
280
Sequence:
MLGQQQQQLYSSAALLTGERSRLLTCYVQDYLECVESLPHDMQRNVSVLRELDNKYQETLKEIDDVYEKYKKEDDLNQKKRLQQLLQRALINSQELGDEKIQIVTQMLELVENRARQMELHSQCFQDPAESERASDKAKMDSSQPERSSRRPRRQRTSESRDLCHMANGIEDCDDQPPKEKKSKSAKKKKRSKAKQEREASPVEFAIDPNEPTYCLCNQVSYGEMIGCDNEQCPIEWFHFSCVSLTYKPKGKWYCPKCRGDNEKTMDKSTEKTKKDRRSR
  
Inhibitor
Name:
BDBM92788
Synonyms:
WAG-005
Type:
Small molecule
Emp. Form.:
C25H30I2NO3
Mol. Mass.:
646.319
SMILES:
CCCCc1oc2ccccc2c1C(=O)c1cc(I)c(OCCC[N+](C)(C)C)c(I)c1
Structure:
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